Animal Models: Use in the Evaluation of Anti-Infective Agents William A. Craig, M.D. University of Wisconsin-Madison

17/06/99

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Table of Contents

Animal Models: Use in the Evaluation of Anti-Infective Agents William A. Craig, M.D. University of Wisconsin-Madison 

Animal Versus In-Vitro Models

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Serum Versus Tissue Concentrations

24-Hr AUC/MIC Required for 1 Log Kill of E.coli in Thighs of Neutropenic Mice

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Pharmacokinetic/Pharmacodynamic Parameters

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Relationship Between Time Above MIC and Efficacy in Animal Infection Models for S. pneumoniae

Time Above MIC vs Efficacy in Acute Otitis Media and Acute Sinusitis

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Relationship Between 24-Hr AUC/MIC and Efficacy of Ciprofloxacin in 64 Patients with Serious Bacterial Infections

PK/PD Parameters: Fluoroquinolones

24-Hr AUC/MIC Ratios for Various Fluoroquinolones Against Streptococcus pneumoniae

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Time above MIC Required for Efficacy of Drug X in Animal Infection Models

Integration of Pharmacokinetics and Pharmacodynamics for Drug X

Dose Determining Studies for Drug Y

24-Hr AUC/MIC Required for Efficacy of Drug Y in Animal Infection Models

Percent Reaching Target AUC/MIC for Static Dose by MIC and Species Following Standard Dose

Percent Expected to Reach Target AUC/MIC When Integrated Over MIC Distribution

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Animal Models for Susceptibility Breakpoint Determinations

Growth of 17 Strains of S. pneumoniae in Thighs of Neutropenic Mice

Effect of Amoxicillin (7 mg/kg) on 17 Strains of S. pneumoniae in Thighs of Neutropenic Mice

Conclusions

Author: William A. Craig (production: Medical Media Production Service) 

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